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Research > Chapter 8012




(2S)-2-Amino-5-chloro-4-hydroxy-5-hexenoic acid chloroamino acid, similar compounds Amanita gymnopus

(2S,1S,2S,3R)-2-(2-carboxy-3-phenylcyclopropyl)glycine potent selective antagonist type 2 metabotropic glutamate receptors

(2S,3S,4R)-2-(Carboxycyclopropyl)glycine potent competitive inhibitor glial neuronal absorption glutamate

(2S,3S,5S)- (2S, 3S, 5R)-5-carboxaldehyde-2,3-diphenyl-1,4-dioxane surrogates optically pure 2,3-O-isopropylideneglyceraldehyde asymmetric synthesis


(2S,4S)-2-amino-4-(2,2-diphenylethyl)pentanedioic acid selective group 2 metabotropic glutamate receptor antagonist

(3)(N,N)-1,8;4,5-naphthalenetetracarboxdiimido-(3)(2,7)pyrenophane (4,4)cyclophane homologue


(3+2) cycloadditions nucleophilic additions aziridines C-C C-N bond cleavage

(3,3)-Sigmatropic ring expansion cyclic thionocarbonates - VOn structure 8-membered thionocarbonates intermediates

(3,3)Sigmatropic ring expansion cyclic thionocarbonates - Highly stereoselective synthesis (Z)- (E)-double bonds controlling chair-like-boat-like transition states (3,3)sigmatropic rearrangement 8-membered thionocarbonates

(3,3)Sigmatropic ring expansion cyclic thionocarbonates - Total synthesis racemic yellow scale pheromone 10-membered thiolcarbonate

(3,3)Sigmatropic ring expansion cyclic thionocarbonates - VRegioselective Wohl-Ziegler bromination 10-membered thiolcarbonates

(3-(4-(4,5-diphenyl-2-oxazolyl)-5-oxazolyl)phenoxy)acetic acid (BMY45778) potent non-prostanoid prostacyclin partial agonist - Influences platelet aggregation, adenylyl cyclase, cAMP levels, protein kinase, iloprost binding


(3-pyridazinamin-3-yl) alpha-aminoacids. facilitated technique preparation phenylalanine proline representatives

(31P)/(1H) nuclear magnetic resonance study mitigating effects GYKI 52466 kainate-induced metabolic impairment perfused rat cerebrocortical slices



(32P)orthophosphate incorporation phospholipids rat liver mitochondria ageing



(Annual Meeting Society Toxicology, Anaheim, California, USA) Immunotoxicity clinical devices

(Annual Meeting diagnosis respiratory allergens Anaheim, California, USA, 1996)



(3H) Aniracetam binds special recognition sites brain membranes

(3H) Clozapine suitable radioligand labelling D-4 dopamine receptors postmortem human brain

(3H) Dopamine absorption platelet storage granules Parkinson's disease

(3H) Hemicholinium-3 binding sites postmortem brains human patients Alzheimer's disease multi-infarct dementia


(3H) Imipramine binding brain samples depressed suicides controls - 5-HT absorption sites compared sites defined desmethylimipramine

(3H) Imipramine binding type I type II alcoholism


(3H) Methoxytetrabenazine. high special activity ligand estimating monoaminergic neuronal integrity

(3H) Neurotensin receptor densities human postmortem brain tissue attained normal schizophrenic persons. An autoradiographic study

(3H) Noscapine binding sites brain - Relationship indoleamines phosphoinositide adenylyl cyclase messenger systems

(3H) Paroxetine binding altered hippocampus frontal cortex caudate nucleus subjects schizophrenia

(3H) Paroxetine binding platelets patients social phobia - Comparison patients panic disorder healthy volunteers

(3H) Phenytoin identifies anticonvulsant-binding domain voltage-dependent sodium channels

(3H) R-Terazosin binds selectively alpha-11-adrenoceptors alpha-2-adrenoceptors-comparison racemic (3H) terazosin (3H)prazosin

(3H) Resiniferatoxin binding human vanilloid (capsaicin) receptor

(3H) Rolipram binding phosphodiesterase activity neuroblastoma N18TG-2 glioma C6Bu-1

(3H) bafilomycin probe transmembrane proton channel osteoclast vacuolar H+-ATPase

(3H) paroxetine binding sites - Brain regional differences psychogenetically selected lines rats

(3H)(+)-7-OH-DPAT (3H)pramipexole binding striatum nucleus accumbens Sprague-Dawley Fischer-344 rats

(3H)(+)-pentazocine binding rat brain sigma-1 receptors

(3H)(+)S 14297:A novel, selective radioligand cloned human dopamine D-3 receptors

(3H)(azidophenyl)ureido taxoid photolabels peptide amino acids 281-304 alpha-tubulin

(3H)(beta-Ala-8)neurokinin A-(4-10). novel, selective radioligand tachykinin NK-2 receptor

(3H)-(+)-pentazocine binding sigma recognition sites human cerebellum

(3H)-(R)-N-6-phenylisopropyladenosine agonist binding solubilized A-1 adenosine receptor bovine epididymal spermatozoa

(3H)-2,3,7,8-TCDD absorption elimination kinetics medaka (Oryzias latipes)

(3H)-L-2-amino-4-phosphonobutyrate labels metabotropic glutamate receptor, mGluR4a

(3H)-MK801 (3H)-NECA binding change administration cyclopentyl adenosine convulsant drug 3-mercaptopropionic acid

(3H)-Noradrenaline release streptolysin-O permeated rat cortical synaptosomes - Enhancement Ca-2+-induced signal


(3H)-RS-45041-190. selective high-affinity radioligand I-2 imidazoline receptors

(3H)-SCH 58261 labelling functional A2A adenosine receptors human neutrophil membranes

(3H)-SR 27897B. selective probe autoradiographic labelling CCK-A receptors brain

(3H)-Thioperamide radioligand the histamine H-3 receptor rat cerebral cortex

(3H)-amino acid absorption metabolic investigations Gigantocotyle explanatum Gastrothylax crumenifer (Digenea - Paramphistomidae)

(3H)-lifarizine high affinity probe inactivated sodium channels

(3H)-monoamine absorption inhibition properties kava pyrones

(3H)-noradrenaline secretion rat cortex synaptosomes perforated Staphylococcus aureus alpha-toxin

(3H)-thyrmidine absorption lipid peroxidation tumor cells embelin cure - An vitro study

(3H)1,3-di(2-tolyl) guanidine binds sigma-2 receptor Jurkat cell membranes, sigma compounds fail effect immunomodulatory events human peripheral blood lymphocytes

(3H)1,3-di-(tolyl)guanidine (3H)(+)pentazocine binding sites rat brain - Autoradiographic visualization putative sigma-1 sigma-2 receptor subtypes

(3H)1-aminocyclopropanecarboxylic acid probe strychnine-insensitive glycine receptors


(3H)2-(2-benzofuranyl)-2-imidazoline. selective high affinity radioligand study rabbit brain imidazoline I-2 receptors

(3H)5,7-dichlorokynurenic acid recognizes binding sites rat cerebral cortex membranes

(3H)5-hydroxytryptamine labels agonist high affinity condition cloned rat 5-HT-4 receptor

(3H)7-Azido-4-isopropylacridone labels Cys159 bovine mitochondrial ADP/ATP-carrier protein

(3H)7-OH-DPAT capable labeling dopamine D-2 D-3 receptors

(3H)7-OH-DPAT labels dopamine D-3 receptors sigma sites bovine caudate nucleus


(3H)8-OH-DPAT labels 5-HT site coupled inhibition phosphoinositide hydrolysis dorsal raphe

(3H)9-Methyl-7-bromoeudistomin D caffeine-like powerful Ca-2+ releaser, binds caffeine-binding sites distinct ryanodine receptors brain microsomes

(3H)A-69024. non-benzazepine ligand vitro vivo investigations dopamine D1 receptors

(3H)A-81988 potent, selective, competitive antagonist radioligand angiotensin AT-1 receptors

(3H)Adenosine transport DDT-1 MF-2 smooth muscle cells - Inhibition metabolites propentofylline

(3H)Adenosine transport rat dorsal brain stem crude synaptosomal preparation


(3H)BQ-123 highly special reversible radioligand endothelin ET-A receptor subtype

(3H)Benzylpempidine radioligand probing putative channel site nicotinic cholinergic receptors

(3H)CGP 39653 binding agonist site N-methyl-D-aspartate receptor modulated Mg-2+ polyamines independently arcaine-sensitive polyamine site

(3H)D-Aspartate binding sites normal human spinal cord motor neuron disease. quantitative autoradiographic study

(3H)DOPA formed (3H)tyrosine living rat brain committed dopamine synthesis

(3H)Dexamethasone binding activity liver microsomes modulated differently 17 alpha-alkylated androgens testosterone vivo

(3H)Dexmedetomidine, alpha-2-adrenoceptor agonist, detects imidazole binding site adult rat spinal cord


(3H)Dizocilpine association kinetics distinguish stimulatory inhibitory polyamine sites N-methyl-D-aspartate receptors

(3H)Dofetilide binding cardiac myocytes - Modulation extracellular potassium


(3H)Dopamine absorption adrenal chromaffin cells mice acute immobilization stress - Difference dark light period

(3H)Forskolin binding cardiac adenylate cyclase guinea pigs chronically infused isoproterenol

(3H)GABA absorption GABA localization mucosal endocrine cells rat stomach colon

(3H)GBR 12935 binding platelets. potential association cytochrome P-450IID6?

(3H)GBR 12935 labels piperazine acceptor site rat prefrontal cortex

(3H)GBR-12935 binding cytochrome P450 human brain

(3H)GBR-12935 binding human cerebral cortex dopamine absorption sites

(3H)Gabapentin label system-L-like neutral amino acid carrier brain


(3H)Homoquinolinate binds subpopulation NMDA receptors binding site


(3H)Inositol hexaphosphate (phytic acid) rapidly absorbed metabolized murine human malignant cells vitro


(3H)L-655,708 ligand selective benzodiazepine site GABA-A receptors alpha-5 subunit

(3H)L-694,247 labels 5-HT-1Dbeta receptor swine caudate membranes

(3H)L-N-G-nitroarginine binding transient focal ischemia NMDA-induced excitotoxicity type I type III nitric oxide synthase null mice

(3H)L-arginine transport and nitric oxide synthase activity in foetal hypothalamic cultures

(3H)LY303870 nonpeptide radioligand NK-1 receptor

(3H)LY341495 highly potent, selective radioligand labeling group II metabotrophic glutamate receptors


(3H)MDL 105,519 binds equal high affinity assembled unassembled NR1 subunits NMDA receptor


(3H)MK-801 binding mRNA NMDAR1 subunit NMDA receptor differentially distributed human rat forebrain

(3H)MK-801 binding asymmetry IMHV area dark-reared chicks reversed imprinting

(3H)MK-801 binding synaptic membranes rat forebrains - Age-related regulation glutamate, glycine spermine

(3H)MK-801 binding well-washed rat brain membranes cessation chronic phencyclidine cure

(3H)N-Methylscopolamine dissociation muscarine receptors affected concentrations allosteric modulators

(3H)Naloxone binding human brain - Alcoholism TaqI A D-2 dopamine receptor polymorphism

(3H)Naloxone binding sites porcine ovarian follicles corpora lutea ovarian cycle

(3H)Nemonapride (3H) spiperone label equivalent numbers D-2 D-3 dopamine receptors range tissues diverse conditions

(3H)PD 140376. highly selective antagonist radioligand cholecystokinin-B/gastrin receptor guinea swine cerebral cortex gastric mucosa

(3H)Paroxetine (3H)citalopram markers human brain 5-HT absorption site. comparison study

(3H)Phorbol 12,13-dibutyrate/PKC binding thoracic spinal cord - No change amyotrophic lateral sclerosis


(3H)QNB displays vivo selectivity m2 subtype

(3H)RS 57639 high affinity, selective 5-HT-4 receptor partial agonist, specifically labels guinea-pig striatal rat cloned (5-HT-4S 5-HT-4L) receptors


(3H)RS79948-197 binding human, rat, guinea swine swine alpha2A-, alpha2B- alpha2C-adrenoceptors. Comparison MK912, RX821002, rauwolscine yohimbine

(3H)Raclopride (3H)spiroperidol binding retinal membranes teleost Eugerres plumieri - Influence light dark adaptation

(3H)Raclopride binding brain tissue subjects schizophrenia - Methodological aspects


(3H)Resiniferatoxin binding swine dorsal horn membranes displays positive cooperativity

(3H)Ryanodine binding sites SR vesicles chicken pectoral muscle

(3H)SCH 58261 selective adenosine A2A receptor antagonist, ligand autoradiographic investigations

(3H)SR 48692, preliminary nonpeptide neurotensin antagonist radioligand - Characterization binding properties proof distinct agonist antagonist binding domains rat neurotensin receptor

(3H)Substrate- cell-specific effects absorption inhibitors human dopamine serotonin transporter-mediated efflux

(3H)Sumatriptan binding sites human brain - Regional-dependent labelling 5-HT-1D 5-HT-1F receptors

(3H)WAY-100635 5-HT-1A receptor autoradiography human brain. comparison (3H)8-OH-DPAT demonstration increased binding frontal cortex schizophrenia


(3H)WIN 35,428 (2-beta-carbomethoxy-3-beta-(4-fluorophenyl)tropane) binding rat brain membranes - Comparing dopamine cell body areas nerve terminal regions


(3H)WIN 35,428 binding human brain

(3H)WIN 35,428 binding dopamine absorption carrier - Influence tonicity buffer composition

(3H)WIN 35,428 binding dopamine absorption carrier - Influence membrane fractionation procedure freezing

(3H)YM-09151-2 (nemonapride) potent radioligand sigma-1 sigma-2 receptor subtypes

(3H)Zolpidem binding alcohol-preferring non-preferring rat brain

(3H)alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) binding anticonvulsant valproate clinically relevant concentrations - An autoradiographic investigation human hippocampus

(3H)bosentan binding human coronary artery - Functional correlates

(3H)bradykinin receptor-binding, receptor-recycling, receptor-internalization B-2 bradykinin receptor murine osteoblast-like cell line MC3T3-E1

(3H)dipyridamole (3H)nitrobenzylthioinosine binding sites human parietal cortex erythrocyte adenosine transporter. comparison

(3H)dofetilide binding - Biological models manifest solely high affinity binding site


(3H)labeled affinity photoaffinity nicotine analogues probing brain nicotinic cholinergic receptors

(3H)nemonapride binding human caudate putamen

(3H)nisoxetine binding sites cat brain - An autoradiographic study

(3H)nisoxetine radioligand noradrenaline reuptake sites - Correlation inhibition (3H)noradrenaline absorption influence DSP-4 lesioning antidepressant treatments

(3H)ouabain binding cultured endothelial cells - Influence cholesterol enrichment

(3H)pBC 264 suitable probe study cholecystokinin-B receptors - Binding characteristics rodent brains comparison (3H)SNF 8702

(3H)propyl-6-azido-beta-carboline-3-carboxylate. photoaffinity label GABA-A-benzodiazepine receptor


(3H)tricyclopinate binding brain muscarinic acetylcholine receptors. comparison (3H)quinuclidinyl benzilate

(3R)-N-(1-(tert-Butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4-benzodiazepin-3-yl)-N-(3-(methylamino)phenyl)urea (YF476). potent orally active gastrin/CCK-B antagonist


(3R,4S)-3-(4-(4-fluorophenyl)-4-hdyroxypiperidin-1-yl)chroman-4,7-diol. conformationally restricted analogue NR2B subtype-selective NMDA antagonist (1S,2S)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidino)-1-propanol

(3R,4S)-3-benzyl-4-bromomethyloxetan-2-one rapid acting alternate substrate inhibitor alpha-chymotrypsin

(3S,4S,5R)-3,4,5-trihydroxy-1-cyclohexene-carboxylic acid Sequoiadendron giganteum

(3SR,4aRS,6SR,8aRS)-6-(1H-Tetrazol-5-yl)decahydroisoquinoline-3-carboxylic acid novel, competitive, systemically active NMDA AMPA receptor antagonist


(3aR,*6aS*)-6a-hydroxy-asymmetric synthesis cyclopenta(b)pyrrole-3a-carboxylate measurement stereostructure NMR spectrum

(4 2) (3 2) cycloaddition reactions 2,3-dideoxy-3-nitro-23-didehydrothymidine ethyl vinyl ether

(4+2) (2+2) cycloaddition reactions 1-(4-methylphenyl) 1-benzyl-1,3-diaza-1,3-butadienes ketenes

(4+2) cycloadditions 2-pyrones benzyne. Application synthesis binaphthyls

(4-(18F)Fluoro-3-iodobenzyl)guanidine potential MIBG analogue positron emission tomography

(4-O-methyl-alpha-D-glucurono)-D-xylan Rudbeckia fulgida, var. sullivantii (Boynton Beadle)


(4fwdarw4)-di(2,3-anhydropentopyranosides) class potential enzyme inhibitors

(51Cr)EDTA measuring total single nephron glomerular filtration rate rat

(5th) International Symposium Work Group Hazards plant-protection products bees ICPBR Programme (Wageningen, Netherlands, October 26-28, 1993)

(6-Maleimidocaproyl)hydrazone doxorubicin-A derivative preparation immunoconjugates doxorubicin

(6-chloro-3-pyridylmethyl-3H)neonicotinoids high-affinity radioligands nicotinic acetylcholine receptors - Preparation NaB-3H-4 LiB-3H-4

(6-oxo-3-pyridazinyl)-benzimidazoles potent angiotensin II receptor antagonists

(6R)-5,6,7,8-Tetrahydro-L-biopterin modulates nitric oxide-associated soluble guanylate cyclase activity rat cerebellum

(6R)-6-(substituted methyl)penicillanic acid sulfones - Novel potent beta-lactamase inhibitors



(7-D-ALA)-angiotensin 1-7 blocks renal actions angiotensin 1-7 anesthetized rat

(7-D-ALA)-angiotensin-(1-7) - Selective antagonism angiotensin-(1-7) rat paraventricular nucleus

(8+2) cycloaddition reactions 2H-cyclohepta(b)furan-2-one acyclic 1,3-dienes. facile bicyclo (5.3.0) ring systems

(8-14C) Inosine metabolism Streptomyces yokosukanensis ATCC 25520

(8-14C)Adenosine (8-14C)inosine metabolism Lepista (Clitocybe) nebularis (Batsch - Fr.) Kummer

(8-Carbon-14) adenosine-5-monophosphate cytokinin biosynthesis germinating corn embryos

(8Z,13Z,20Z)-Strobilinin (7Z,13Z,20Z)-felixinin - Novel furanosesterterpene tetronic acids marine sponges genus Ircinia

(99mTc)tricine. precursor complex radiolabeling hydrazinonicotinate protein conjugates

(9;11) (p22;q23) translocation blastic phase chronic myeloid leukemia

(A,G)-oligonucleotides form extraordinary stable triple helices critical R cntdot Y sequence murine c-Ki-ras promoter inhibit transcription transfected NIH 3T3 cells

(ATT) trinucleotide repeats antithrombin gene determining origin repeated mutations

(Adeno)tonsillectomy children

(Ala-6,D-Trp-8) Galanin(1-15)ol potent galanin antagonist insulin release

(Ala4)Surfactin isoform Bacillus subtilis studied mass NMR spectroscopies


(Aminoalkyl)indole isothiocyanates potential electrophilic affinity ligands brain cannabinoid receptor

(Aminomethyl)phosphonate derivatives oligonucleotides


(Anguilliform fishes Reunion (Indian Ocean). Portrayal species


(Apo)lipoproteinConcentrations Birth Preliminary Days Months Life-Investigations Distribution Serum Levels Predictive Value Measurements Made Time

(Arg-8) Vasopressin-induced responses human extracted coronary artery - Influences non-peptide receptor antagonists

(Arg-8)Vasotocin excites neurones dorsal vagal complex vitro - Proof effect class(es) CNS receptors

(Arg15, Arg21) VIP - Evaluation biological activity localization breast cancer tumors


(Aryloxy)alkylamines selective human dopamine D4 receptor antagonists - Potential antipsychotic agents

(Aryloxy)aryl semicarbazones similar compounds. class anticonvulsant agents possessing high activity maximal electroshock screen

(Aryloxy)methylsilane derivatives cholesterol biosynthesis inhibitors - Synthesis hypocholesterolemic activity class squalene epoxidase inhibitors

(Boro)hydride techniques trace element speciation





(CT)-n (GT)-n microsatellites. class genetic markers Salmo trutta L. (brown trout)


(CTG)-n triplet mutation phenotype manifestations myotonic dystrophy patients

(Ca+Mg)ATPase calcium influx erythrocytes patients idiopathic hypercalciuria

(Ca-2+) Modulates ratio cyclooxygenase lipoxygenase metabolism arachidonic acid homogenates hippocampal astroglial cultures



(Ca-2+)-i pH-in homeostasis Kaposi sarcoma cells

(Ca-2+)-i protein kinase C vasopressin-induced prostacyclin ANP release rat cardiomyocytes

(Ca-2+)-i arising individual guinea-pig chromaffin cells answer receptor agonists relationship catecholamine secretion perfused adrenal gland



(Ca-2+)-i human heart failure. review discussion current areas controversy

(Ca-2+)-i rat afferent arteriole constriction measured confocal fluorescence microscopy



(Ca-2+)-i oscillations (Ca-2+)-i waves rat megakaryocytes

(Ca-2+)-i oscillations rat chromaffin cells - Frequency amplitude modulation Ca-2+ InsP-3

(Ca-2+)-i oscillations single rat glioma cells stimulated thrombin activation cell surface receptors


(Ca-2+)-i oscillations stimulated bradykinin rat glioma cells Ca-2+ store-dependent Ca-2+ influx controlled cell volume membrane potential

(Ca-2+)-i oscillations stimulated muscarinic stimulation airway smooth muscle cells - Receptor subtypes correlation mechanical activity


(Ca-2+)-i regulation glutamate receptor agonists cultured chick retina cells

(Ca-2+)-i signaling pregnant human myometrium

(Ca-2+)-i transients hypertensive postinfarction myocytes


(Ca-2+)-i-sensitive, IP-3-independent Ca-2+ influx smooth muscle rat vas deferens revealed procaine

(Ca-2+)-i-transients actin polymerization human neutrophils stimulation GRO-alpha complement fragment C5-a

(Ca2+)i-reducing effect cAMP rat pancreatic beta-cells - Involvement thapsigargin-sensitive stores

(Carboxyalkyl)benzyl propargyl ethers selective inhibitors leukocyte-type 12-lipoxygenases

(Carboxyalkyl)pyrroles human plasma oxidized low-density lipoproteins

(Cis)-preference N,N-dimethyl-N,N-diphenylguanidine guanidinium salt. Construction water-soluble aromatic layered formation


(Co) variance constituent estimates milk composition traits Sarda dairy sheep bivariate animal model

(Co)variance constituent estimation yield traits diverse lactations animal model

(Conference on) Environmental Pollution Child Health in ern Europe, (Sosnowiec, Poland; May 8-10, 1996; School Public Health, University Albany, State University Novel York; Institute Occupational Medicine Environmental Health, Sosnowiec, Poland; National Institute Environmental Health Sciences (NIEHS); WHO-European Centres Environment Health; Fogarty International Center, National Institutes Health)

(Corrected reprinted volume 78, pages 319-333, 1998) - Development, progression, androgen-dependence prostate tumors probasin-large T antigen transgenic mice. model prostate cancer

(Cys(O-2NH-2)-2)enkephalin analogues dalargin - Selectivity delta-opioid receptors

(D)-penicillamine increases hepatic oxalate production resulting hyperoxaluria

(D-Ala, D-Leu) enkephalin reduces binding GTP hippocampal membranes


(D-Arg-1, D-Phe-5, D-Trp-7,9, Leu-11) agent P induces apoptosis lung cancer cell lines vitro

(D-Arg-1, D-Phe-5, D-Trp-7,9, Leu-11) agent P inhibits growth human cell lung cancer xenografts vivo

(D-Arg-1,D-Trp-5,7,9,Leu-11)Substance P. potent inhibitor signal transduction growth vitro vivo cell lung cancer cells



(D-Leu-2)deltorphin 17 amino acid opioid peptide skin Brazilian hylid frog, Phyllomedusa burmeisteri

(D-Pen-2, D-Pen-5)enkephalin delta opioid agonist, reduces endogenous aluminum content rat nervous scheme

(D-Pen-2,5)enkephalin glutamate regulate expression delta-opioid receptors rat cortical astrocytes

(D-Pro-5) corticotropin-releasing factor analogs selective agonists corticotropin-releasing factor receptors

(D-TRP-32) neuropeptide Y. competitive antagonist NPY rat hypothalamus

(D-pen-2-D-pen-5)enkephalin delta opioid agonist, intracerebroventricularly mouse produces antinociception mediation spinal GABA receptors

(DIS)respect black mortality

(Daily activity pattern behavior Thomas leaf monkey Presbytis thomasi Collet 1892) Ketambe forest, Gunung Leuser National Park,east Aceh

(Delphinidin 3-gentiobiosyl) (apigenin 7-glucosyl) malonate flowers Eichhornia crassipes


(Dextro)-13-alpha-(4-hydroxytigloyloxy)lupanine Ormosia krugii


(Dextro)-HA 966 partial agonist glycine site coupled NMDA receptors, blocks formalin-induced pain mice

(Dextro)-hitachimycin - Stereochemistry conformational examination

(Dipropylamino)-tetrahydronaphthofurans:ly acting serotonin agonists dopamine agonists-antagonists

And (Z) 5-fluoroolefin carbocyclic nucleosides - Influence olefin geometry inhibition S-adenosyl-L-homocysteine hydrolase

And (Z)-3-styrylpiperidines sigma ligands

(E)- (Z)-7-arylidenenaltrexones - Synthesis opioid receptor radioligand displacement assays

(E)-(arylmethyleneaminoxy)acetamides analogues neuroleptic benzamides - Synthesis D-2-dopaminergic binding affinity

(E)-(methyloxyimino)acetamides analogues neuroleptic benzamides - Synthesis D-2-dopaminergic binding affinity

(E)-1-(heterocyclyl cyclohexyl)-2-(1,3,7-trisubstituted (xanthin-8-yl)) ethenes A-2a adenosine receptor antagonists

(E)-1-Alkyl-(2-(1H-azol-2-yl)vinyl)pyridinium salts - Theoretical analysis, synthesis assessment interaction choline acetyltransferase


(E)-2-hexenal induce Botrytis cinerea growth vitro strawberries vivo storage

(E)-2-hexenal-induced DNA damage structure cyclic 1,N-2-(1,3-propano)-2-deoxyguanosine adducts mammalian cells

(E)-3((((6-(2-Carboxyethenyl)-5-((8-(4-methoxyphenyl)octyl)oxy)-2-pyridinyl)-methyl)thio)methyl)benzoic acid similar compounds - High affinity leukotriene B-4 receptor antagonists

(E)-3-(2-(N-phenylcarbamoyl)vinyl)pyrrole-2-carboxylic acid derivatives - class glycine site antagonists

(E)-3-(6-(((2,6-dichlorophenyl)thio)methyl)-3-(2-phenylethoxy)-2-pyridinyl)-2-propenoic acid. high-affinity leukotriene B-4 receptor antagonist oral antiinflammatory activity

(E)-3-Tridecen-2-one, antibiotic interdigital glands black-tailed deer Odocoileus hemionus columbianus

(E)-4-(2-((3-(indol-5-yl)-1-oxo-2-butenyl)amino)phenoxy)butyric acid derivatives. class steroid 5-alpha-reductase inhibitors rat prostate. 1

(E)-4-hydroxy-2-nonenal involved pathogenesis Parkinson's disease

(E)-5,6-Didehydro-6-deoxy-6-fluorohomoadenosine. substrate measures hydrolytic activity S-adenosylhomocysteine hydrolase

(E)-5-(2-bromovinyl)-2-deoxyuridine inhibition macropodid herpesvirus 1 vitro

(E)-5-Tosyl-4-pentenamide. vinyl sulfone one-pot general synthesis indolizidine derivatives

(E)-8-benzylidene derivatives 2-methyl-5-(3-hydroxyphenyl) morphans - Highly selective ligands sigma-2 receptor subtype

(E)-bis-1,2-(tributylstannyl)ethylene staple synthetic advance taxol

(E)-enolbutyryl-UDP-N-acetylglucosamine mechanistic probe UDP-N-acetylenolpyruvylglucosamine reductase (MurB)

(E)4-(4-N,N-dimethylaminophenyl)but-3-en-2-one (DMAP) cure inhibits radiation-induced micronucleus structure bone marrow BALB/c mice

(E,Z)- (E,E)-10,12-hexadecadienals, major components female sex pheromone cotton leaf-roller, Notarcha derogata (Fabricius) (Lepidoptera - Pyralidae)


(ECTO) nucleotidase kinetics observed 31P-NMR spectroscopy - Resolution signals

(Enantio-)separation phenoxy acid herbicides capillary zone electrophoresis


(European Charcot Foundation Symposium Body fluid markers monitor multiple sclerosis - The assays challenges, Madrid, Spain, October 24, 1997)

(Fe(PMA))-n positive (n equals 1,2) - Good models iron bleomycins examples mononuclear non-heme iron complexes significant oxygen activation capabilities

(Flowers visited syrphids (Diptera - Syrphidae) mesophilous forest Campinas, SP)

(Fluorocyclopropyl)quinolones - Synthesis stereochemical structure-activity relationships chiral 7-(7-amino-5-azaspiro(2.4)heptan-5-yl)-1-(2-fluorocyclopropyl)quinolone antibacterial agents

(G586V) Substitutions alpha-1 alpha-2 chains collagen. I - Influence alpha-chain stoichiometry phenotype osteogenesis imperfecta?


(GT)-n repetitive tracts affect stages RecA-promoted recombination

(GTG).5 distinction diverse isolates nematode Caenorhabditis elegans

(Galacto)lipid export envelope thylakoid membranes intact chloroplasts. A general process key function envelope establishment lipid asymmetry thylakoid membranes

(Glyco)-protein drug carriers intrinsic therapeutic activity - The concept dual targeting


(H)GBR 12935 binding human platelet membranes sensitive piperazine derivatives dopamine absorption inhibitors



(Helicobacter-pylori atrophic gastritis

(His)C&e-H cntdot cntdot O=C hydrogen bond active sites serine hydrolases

(Hydroxyethyl) sulfonamide HIV-1 protease inhibitors - Identification 2-methylbenzoyl moiety P-2


(Imidazolylphenyl)pyrrol-2-one inhibitors cardiac cAMP phosphodiesterase

(In)curability breast cancer. 30-year report series 3933 cases

(Iodine)-iodomelatonin-binding sites bursa Fabricius birds - Binding characteristics, subcellular distribution, diurnal variations age investigations

(Iodine-125) neurokinin A labels pharmacologically distinct populations NK-2 binding sites hamster rabbit urinary bladder



(K+)out accelerates inactivation of Shal-channels responsible for A-current in rat CA1 neurons

(L-Ala-3)DPDPE. enkephalin analog unique opioid receptor activity profile. Further proof delta-opioid receptor multiplicity

(Latent) transforming growth factor beta liver parenchymal cells, injury-dependent release, paracrine effects rat hepatic stellate cells

(Leu)enkephalin enhances active avoidance conditioning rats mice

(Leu-31,Pro-34) neuropeptide Y (NPY), NPY 20-36, produces discriminative stimulus effects related NPY induces food intake


(Leu-8) des-Arg-9-bradykinin inhibits angiogenic influence bradykinin interleukin-1 rats

(Leucine-5)enkephalin-like immunoreactive amacrine cells nicotinic excitatory control darkness chicken retina

(Levo)-penbutolol blocker of 5-HT-1A receptor-mediated responses

(Lys(-2)-Arg(-1))endothelin-1 solution formation two-dimensional 1H-NMR - Possible involvement electrostatic interactions native disulfide bridge formation biological activity decrease

(Lys(B28), Pro(B29))-human insulin - Influence injection time postprandial glycemia

(Lys(B28), pro(B29))-Human insulin. rapidly absorbed analogue human insulin

(MPR-14)-rADM(14-50) analog adrenomedullin, possesses potent vasodilator activity hindlimb vascular bed cat

(Melle-4)cyclosporin natural cyclosporin anti-HIV activity - Structural elucidation, biosynthesis biological properties


(Met-5)enkephalin delta-2-opioid receptors spinal cord involved cold water swimming-induced antinociception mouse


(Methyl-carbon-11)thymidine vivo determination cell proliferation

(N-methyl-3H) methylphenazepam. ligand benzodiazepine receptors

(N-methylnorleucine-(28,31))cholecystokinin-(26-33) (SNF 8702) activity cloned rat CCK-B receptor

(NAD+)/(NADH) redox-state metabolites freeze-clamped livers rats fed casein gelatin diets

(NANP) 19-5.1. malaria vaccine field experiment Nigerian children

(NH-4+ + Na+)-activated ATPase facultatively anaerobic alkaliphile, Amphibacillus xylanus

(Non)issues infinite regress modeling motor behavior

(O-ethyl 14C)phenacetin O-deethylase activity human liver microsomes

(O-methyl 14C)naproxen O-demethylase activity human liver microsomes - Proof involvement cytochrome P4501A2 P4502C9/10

(O-methyl-11C)beta-CIT-FP potential radioligand quantitation dopamine transporter - Preparation, autoradiography, metabolite studies, positron emission tomography examinations


(Os(bpy)-2(PVI)-10Cl)Cl polymer-modified carbon fiber electrodes electrocatalytic oxidation NADH

(PRO-9)SP (pGLU-6, PRO-9)SPO(6-11) interact diverse receptors guinea-pig ileum demonstrated SP antagonists

(PSI) (URE3) yeast prions

(Phe-22)-big endothelin-1(19-37). potent inhibitor endothelin-converting enzyme

(Phe1PSI(CH2-NH)Gly2) nociceptin-(1-13)-NH2 acts agonist orphanin FQ/nociceptin receptor vivo

(Phe1psi(CH2-NH)Gly2)-nociceptin-(1-13)NH2 proposed antagonist nociceptin receptor, potent stable agonist rat spinal cord

(Phe1psi(CH2-NH)Gly2)nociceptin-(1-13)-NH2 agonist nociceptin (ORL1) receptor

(Phe21)big endothelin-1(18-34) (Ala31)big endothelin-1(18-34) inhibit human endothelin-converting enzyme-1 (ECE-1) expressed CHO-K1 cells diverse fashion

(Pheo)melanin photosensitizes UVA-induced DNA damage cultured human melanocytes

(Pinless Fixation. Part II) - Documentation

(Piperidinylalkoxy)chromones - New antihistamines antagonistic activity leukotriene D-4

(Pre-)disposition, variation fitness illustrated evolutionary forming inflorescence blossoms


(Pro-34) peptide YY Y-1-selective agonist peptide YY/neuropeptide Y receptors

(Pro11,D-Ala12)angiotensin I fast onset vasoconstrictor activity cat



(R) (S) RS 56532 - Mixed 5-HT-3 5-HT-4 receptor ligands opposing enantiomeric selectivity

(R)(+)-N-Propargyl-1-aminoindan (rasagiline) derivatives - Highly selective potent inhibitors monoamine oxidase B

(R)- (S)-8-acetyl-2-(dipropylamino)tetralin (LY-41) - Two 5-HT-1A receptor agonists

(R)-(+)-2(((3-(morpholinomethyl)-2H-chromen-8-yl)oxy)methyl)morpholine methanesulfonate. selective rat 5-hydroxytryptamine1B receptor antagonist

(R)-(+)-N-(3-(5-((4-fluorophenyl)methyl)-2-thienyl)-1-methyl-2-propynyl)-N-hydroxyurea (ABT-761) second-generation 5-lipoxygenase inhibitor

(R)-(+)-menthofuran potent, mechanism-based inactivator human liver cytochrome P450 2A6

(R)-(dextro)- (S)-(levo)-5-ethyl-5-methyl-1,3-dioxolane-2,4-dione reagents direct preparation alpha-hydroxy-alpha-methylbutyrate esters - Assignment absolute configuration alpha-acetoxy-a-methylbutyrate ester side chain quassimarin total synthesis

(R)-(levo)-(E)-2,6-dimethyl-3,7-octadiene-2,6-diol 6-O-beta-D-glucopyranoside - Natural precursor hotrienol lulo fruit (Solanum vestissimum D.) peelings

(R)-1,2,3,4-tetrahydro benzothieno (2,3-c) pyridines - New optically active compounds strong 5-HT-1A receptor binding ability exhibiting anticonflict activity lessening memory impairment

(R)-11-hydroxy-and (R)-11-hydroxy-10-methylaporphine - Synthesis, pharmacology, modeling D-2A 5-HT-1A receptor interactions


(R)-2-Octeno-delta-lactone volatiles produced Lasiodiploida theobromae

(R)-3-(6-chloro-1-isopropylbenzimidazole-4-carboxamido)quinuclidine. high affinity ligand (R)-zacopride binding site

(R)-5-Fluoro-5,6-dihydrouracil - Kinetics oxidation dihydropyrimidine dehydrogenase hydrolysis dihydropyrimidine aminohydrolase


(R)-Alpha-methylhistamine inhibits ethanol-induced gastric lesions rat - Involvement histamine H-3 receptors?

(R)-Isovaline Homo-Peptides Adopt Left-Handed 3-10-Helical Structure

(R)-Thionisoxetine potent selective inhibitor of peripheral norepinephrine absorption

(R)-and (S)-coclaurine bark Peumus boldus


(R)-methanandamide, anandamide, substitutes DELTA-9-THC drug-discrimination procedure

(R)-prechrysophanol Aloe graminicola

(R)salsolinol N-methyltransfer activity increases Parkinsonian lymphocytes

(R,R)-2,2-(1,2-ethanediylbis(imino(1-methyl-2,1-ethanediyl)))-bis(5-nitro-1H-benz(de)isoquinoline-1,3-(2H)-dione) dimethanesulfonate (DMP 840) bis-naphthalimide potent nonselective tumoricidal activity vitro

(R,S)-alpha-Amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) receptors mediate calcium-dependent inhibition metabotropic glutamate receptor-stimulated structure inositol 1,4,5-trisphosphate

(R,S)-alpha-methyl-4-carboxyphenylglycine (MCPG) blocks spatial learning rats long-term potentiation dentate gyrus vivo

(R,S)-alpha-methyl-4-carboxyphenylglycine (MCPG) fails block long-term potentiation urethane anaesthesia vivo

(R-p)- (S-p)-8-piperidino-adenosine 3,5-(cyclic)thiophosphates discriminate completely site A B regulatory subunits cAMP-dependent protein kinase type I II

(R-p)-cAMPS inhibits cAMP-dependent protein kinase blocking cAMP-induced conformational transition

(RS)-2-chloro-5-hydroxyphenylglycine (CHPG) activates mGlu-5, mGlu-1, receptors expressed CHO cells potentiates NMDA responses hippocampus

(RS)-alpha-Methyl-4-carboxyphenylglycine inhibits long-term potentiation function frequency stimulation rat dentate gyrus vitro

(RS)-alpha-methyl-4-carboxyphenylglycine (MCPG) block theta burst-induced long-term potentiation region CA1 rat hippocampal

(Racemic) baclofen sensitive scopolamine-induced short-term memory deficits mice

(Racemic)-(N-alkylamino)benzazepine analogs - New dopamine D-1 receptor antagonists

(Racemic)-(Z)-2-(aminomethyl)-1-phenylcyclopropanecarboxamide derivatives prototype NMDA receptor antagonists

(Racemic)-1-Azabicyclo(2.2.1)heptane-3-one, O-(3-methyl-5-aryl-2-penten-4-ynyl)oximes - Potent muscarinic agonists

(Racemic)-3-(4-(2-dimethylamino-1-methylethoxy)-phenyl)-1H-pyrazolo(3,4-b)pyridine-1-acetic acid (Y-25510) stimulates production IL-1-beta IL-6 degree messenger RNA expression cultured human monocytes

(Racemic)-7-Deazacarbovir compound potential anti-HIV anti-HCMV properties

(Racemic)-7-deazaaristeromycin lacking hydroxymethyl substituent

(Racemic)-8-oxohypecorinine Hypecoum procumbens var. glaucescens

(Racemic)-CP-96, 345, NK-1 receptor antagonist, local anaesthetic-like effects mammalian sciatic nerve preparation


(Racemic)-Kavain inhibits veratridine-activated voltage-dependent Na+-channels synaptosomes prepared rat cerebral cortex

(Racemic)-govadine (Racemic)-THP, tetrahydroprotoberberine alkaloids, selective alpha-1-adrenoceptor antagonists vascular smooth muscle cells

(Racemic)-tamsulosin, alpha-1A-adrenoceptor antagonist, inhibits positive inotropic influence accumulation inositol phosphates rabbit heart

(Racemic)11-Amino-2,6-dimethyl-1,2,3,4-tetrahydro-6H-quinindolin-1-one GABA-A modulator potential anxiolytic activity

(Racemic)CPP, NMDA receptor antagonist, blocks induction commissural-CA3 LTP anesthetized rat


(Rp)-8-pCPT-cGMPS cGMP-dependent protein kinase inhibitor

(Ru-2-II(ttha)(H-2O)-2)-2- fast NO scavenger (ttha-6- equals triethylenetetraminehexaacetate)

(S) Oxazepam glucuronidation inhibited ketoprofen substrates UGT2B7

(S)- (R)-(carbon-11) nicotine metabolite (R/S)-(carbon-11) cotinine - Preparation, metabolite investigations vivo distribution human brain PET

(S)- (R)-8-(di-n-propylamino)-6,7,8,9-tetrahydro-3H-benz(e)indole-1-carbaldehyde. class orally active 5-HT-1A-receptor agonists

(S)-(+)-1-methyl-2-(6,7-dimethoxy-2,3-naphthalimido) ethyl trifluoromethanesulfonate fluorescence chiral derivatizing reagent carboxylic acid enantiomers high-performance liquid chromatography

(S)-(+)-4,4,4-trifluoro-3-(indole-3-)butyric acid fluorinated plant growth regulator

(S)-(dextro)-ipsdienol - Interspecific inhibition Ips latidens (LeConte) Ips pini (Say) (Coleoptera - Scolytidae)

(S)-1-(3-hydroxy-2-(phosphonylmethoxy)propyl)cytosine (Cidofovir) - Results phase I/II study antiviral nucleotide analogue

(S)-1-(3-hydroxy-2-phosphonylmethoxypropyl)cytosine (HPMPC) inhibits HIV-1 replication epithelial cells, T-lymphocytes

(S)-13-((Dimethylamino)methyl)-10,11,14,15-tetrahydro-4,9:16,21-dimetheno-1H,13H-dibenzo(e,k)pyrrolo(3,4-h)(1,4,13)oxadiazacyclohexadecene-1,3(2H)-dione (LY333531) similar analogues - Isozyme selective inhibitors protein kinase C-beta

(S)-13-hydroxygeranylgeraniol-derived furanoditerpenes Bifurcaria bifurcata

(S)-2-Amino-1,3-propanediol-3-phosphate-carrying diradylglyceroglycolipids - New major membrane lipids Clostridium innocuum

(S)-3,7-dimethyl-5-octene-1,7-diol similar oxygenated monoterpenoids petals Rosa damascena Mill



(S)-4-Carboxy-3-hydroxyphenylglycine, antagonist metabotropic glutamate receptor (mGluR)1a agonist mGluR2, protects audiogenic seizures DBA/2 mice

(S)-4-amino-5-chloro-3-iodo-2-methoxy-N-(1-azabicyclo(2.2.2)oct-3-yl)benzamide (TRIZAC) high-affinity ligand 5-HT-3 receptor

(S)-4-carboxy-3-hydroxyphenylglycine activates phosphatidylinositol linked metabotropic glutamate receptors diverse brain regions neonatal rat

(S)-5,7biphyscion 8-glucoside Cassia torosa

(S)-5-fluorowillardiine-mediated neurotoxicity cultured murine cortical neurones occurs AMPA kainate receptors

(S)-9-(3-hydroxy-2-phosphonylmethoxypropyl)adenine ((S)-HPMPA). purine analogue trypanocidal activity vitro vivo

(S)-C-alpha-ethyl, C-alpha-benzylglycine ((S-)-alpha-Et)Phe) peptides fold left-handed helical structures

(S)-Emopamil attenuates acute reduction regional cerebral blood flow experimental brain injury

(S)-Emopamil reduces brain edema collagenase-induced hemorrhage rats


(S)-Homo-AMPA special agonist mGlu6 subtype metabotropic glutamic acid receptors

(S)-Linalyl, 2-phenylethyl, benzyl disaccharide glycosides extracted aroma precursors oolong tea leaves

(S)-UH301, A silent 5-HT-1A receptor antagonist, enhances plasma corticosterone levels rat

(S)-WAY 100135 5-HT-1A receptor antagonist, prevents impairment spatial learning attributable intrahippocampal scopolamine


(S)-cis-2-amino-5-chloro-4-pentenoic acid fungus Amanita vergineoides

(S)-form alpha-methyl-N(alpha)-phthalimidoglutarimide, (R)-form, enhanced phorbol ester-induced tumor necrosis factor-alpha production human leukemia cell HL-60 - Implication optical resolution thalidomidal effects

(S)-ketamine-renaissance substance?

(S)-spiro((1,3-diazacyclopent-1-ene)-5,2-(7-methyl-1,2,3,4-tetrahydronaphthalene)) - Resolution, stereospecific synthesis, pharmacological characterization partial alpha-adrenergic agonist

(S,S)- (S,R)-1-(18F)fluorocarazolol, ligands visualization pulmonary beta-adrenergic receptors PET




(Sp)-8-chloroadenosine 3,5-cyclophosphate stimulated differentiation human leukemia HL-60 cells

(Stearyl, Norleucine-17) VIP hybrid antagonizes VIP receptors non-small cell lung cancer cells


(The Sixth Sandoz-Keystone Symposium Blood Cell Bone Marrow Transplants, Keystone, Colorado, USA, January 15-21, 1996)

(Tibouchina sect. Pleroma (D.Don) Cogn. (Melastomataceae) Sao Paulo state)

(Trifluoromethyl)lumazine derivatives 19F NMR probes lumazine protein

(Tritiated) p-aminoclonidine (tritiated) idazoxan label diverse populations imidazoline sites rat kidney

(Turf) transurethral radiofrequency heating benign prostatic hyperplasia temperatures Thermex II - Clinical experience

(Tyr-1)-nociceptin, nociceptin analog, decreases systemic arterial pressure naloxone-insensitive mechanism rat

(Tyr-5)didemnin B (D-Pro-4)didemnin B; natural didemnins modified macrocycle

(Tyr1)-nociceptin naloxone-insensitive vasodilator activity hindquarters vascular bed rat

(U-13C)glutamate metabolism astrocytes hypoglycemia hypoxia

(U-13C)glutamate metabolism in rat brain mitochondria reveals malic enzyme activity

(URE3) altered URE2 protein - Proof prion analog Saccharomyces cerevisiae

(Volynites Ljashenko, 1957 fauna Lower Devonian Cantabrian Mountains (NW Spain)

(Z)- (E)-2-(hydroxymethyl)cyclopropylidene)methyladenine -guanine, nucleoside analogues broad-spectrum antiviral activity

(Z)-10-Heptadecen-2-one 2-tridecanone biosynthesis (1-carbon-14) acetate Drosophila buzzatii


(Z)-3-(4-Bromophenyl)-3-(3-Pyridyl)allylamine substrate investigations myeloperoxidase activity

(Z)-3-hexenyl-beta-D-glucopyranoside fresh tea leaves precursor green odor

(Z)-4-Tridecenal pheromonally active air oxidation product series (Z,Z)-9,13 dienes Macrocentrus grandii Goidanich (Hymenoptera - Braconidae)


(Z)-selective beta-bromination N-formyl-alpha,beta-dehydroamino acid esters




(alpha-S, Z-1R, 3R)-(4,4-tritiated) cyhalothrin -(4, 6-tritiated)4-fluorocyhalothrin - Synthesis candidate pyrethroid radioligands sodium channel


(cis)-3-Methyl-1,5-benzothiazepine-4-ones - Potent analogs calcium channel blocker diltiazem

(des His-1, des Phe-6, Glu-9)Glucagon amide. newly designed pure glucagon antagonist

(eta-5-Cyclopentadienyl)metal Tricarbonyl Pyrylium Salts - New Reagents Specific Conjugation Proteins Transition Organometallic Labels

(gamma-35S)GTP autoradiography region-specific detection muscarinic receptor-dependent G-protein activation chick optic tectum

(i,i+4) ion pairs stabilized helical peptides derived smooth muscle caldesmon



(levo)-Deprenyl (Selegiline) devoid amphetamine-like behavioural effects rats


(methyl-3H)Thymidine (3H)leucine incorporation Vibrio spp. grown nutrient-limited continuous cultures


(n-3) Polyunsaturated fatty acids modulate expression functionally molecules human monocytes vitro

(n-3) (n-6) PUFA biochemical markers developmental stages brine shrimp developing 'dumpy' 'slender' adults

(omega-(Adenosin-5-O-yl)alkyl)cobalamins mimicking posthomolysis intermediate coenzyme B-12-dependent rearrangements - Kinetic studies methylmalonyl-CoA mutase


(racemic)-3-(4-(N,N-dimethylamino)cinnamyl)benzazepine analogs - New dopamine D-1 receptor antagonists

(racemic)-Gelliusines A B, diastereomeric brominated tris-indole alkaloids deep water Caledonian marine sponge (Gellius Orina sp.)

(racemic)-Kavain inhibits veratridine- KCl-induced increase intracellular Ca-2+ glutamate-release rat cerebrocortical synaptosomes

(racemic)-trans-2-(3-methoxy-4-(4-chlorophenylthioethoxy)-5-(N-methyl-N-hydroxyureidyl)methylphenyl)-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran (CMI-392) potent dual 5-lipoxygenase inhibitor platelet-activating factor receptor antagonist

(s)-Aspartate semi-aldehyde - Synthetic structural investigations

(s-4dU)-35. novel, highly potent oligonucleotide inhibitor human immunoinsufficiency virus type 1 reverse transcriptase

+Gz acceleration affects trace minerals zinc, copper, chromium serum urine humans

+Gz-induced neck injuries royal Australian Air Force fighter pilots

+P5(D1S3309E) target binding site Wilms tumour suppressor 1(WT1) gene, maps human chromosome 1q21 fwdarw q22

,4-diacylpiperazine-2-(S)-((N-aminoalkyl)carboxamines) novel, potent agent P receptor antagonists


-308 tumor necrosis factor (TNF) polymorphism survival severe sepsis unrelated lipopolysaccharide inducibility human TNF promoter


-ffect postweaning nutritional environmental restrictions discrimination learning albino rats


-n vitro measurement creatine kinase substrate fluxes 31P-nuclear magnetic resonance


0-IIb type superficial esophageal carcinoma - For preliminary time recognized chromoendoscopy iodine staining, report case

0.05 percent clobetasol 17-propionate cream ointment 0.1 percent triamcinolone acetonide preparations increase skin surface roughness. potential dissociation unwanted epidermal dermal effects

0.125 percent ropivacaine related 0.125 percent bupivacaine labor analgesia patient-controlled epidural infusion

0.15 mg Clonidine oral premedication surgery retrobulbar anesthesia

0.25 percent chlorhexidine gluconate gel. protective topical microbicide


0.3 percent ciprofloxacin ophthalmic ointment cure bacterial keratitis

0.45 percent saline 5 percent dextrose water, 0.9 percent saline 5 percent dextrose 0.9 saline, worsen brain edema hours closed head trauma rats

013 (CD99) positivity hematologic proliferations correlates TdT positivity

0N0-4007 synthetic lipid A derivative, induces differentiation rat myelomonocytic leukemia cells vitro vivo



1 (2)gl gene regulates late expression segment polarity genes Drosophila

1 Acyl-2 acetyl-sn-glycero-3 phosphocholine decreases vulnerability low-density lipoprotein oxidative modification copper ions, monocytes endothelial cells

1 X ED-90 dose rocuronium bromide - Tracheal intubation conditions time-course effect

1 kb lactase-phlorizin hydrolase promoter directs post-weaning decline intestinal-specific expression transgenic mice

1,2-seco-2,3-dideoxynucleoside analogues - Synthesis antiviral assessment racemic trans-((1,5-dihydroxy-3,4-methylenyl-pent-2-oxy)methyl) nucleosides

1,4-Trans-(14C)-abscisic acid diol. major product R-(2-14C)-mevalonic acid metabolism extracts Citrus sinensis exocarp

1-(2-phenyl-ethylene)-ditryptophenaline dimeric diketopiperazine Aspergillus flavus

1-Acetoxychavicol acetate superoxide anion generation inhibitor potently inhibits tumor promotion 12-O-tetradecanoylphorbol-13-acetate ICR mouse skin

1-Hydroxyeugenol- coniferyl alcohol derivatives effective inhibitors 5-lipoxygenase Cu-2+-mediated density lipoprotein oxidation - Proof dual mechanism

1-acetoxychavicol acetate inhibitor phagocytosis macrophages

1,000 consecutive ultrasounds blunt abdominal trauma

1,1-Dicyano-2-substituted ethylenes. class glucose absorption inhibitors antifilarial chemotherapy


1,1-Ethylidenebis(L-tryptophan) contaminant implicated L-tryptophan eosinophilia myalgia syndrome, suppresses mRNA expression hypothalamic corticotropin-releasing hormone Lewis (LEW/N) rat brain


1,1-ethylidenebis (L-tryptophan), impurity L-tryptophan eosinophilia-myalgia syndrome, stimulates type I collagen gene expression human fibroblasts vitro

1,1,2,2-Tetrachloroethane-induced early decrease dolichol levels rat liver microsomes Golgi apparatus

1,1,3,3-tetraisopropyldisiloxane-1,3-diyl (TIPS) migration facilitates one-pot structure enantiomerically pure methyl 2,3-epoxy-D-xylonate


1,1-Bisphosphonate squalene synthase inhibitors - Interplay isoprenoid subunit diphosphate surrogate



1,1-Dinitroethyl substituted furoxans. class vasodilators inhibitors platelet aggregation

1,1-Diphenoxy-2-(phenylsulfonyl)cyclopropane furan ann